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Home > Products >  PF-06821497

PF-06821497 CAS NO.1844849-10-0

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  • Product Details

Keywords

  • 1(2H)-Isoquinolinone, 5,8-dichloro-2-((1,2-dihydro-4-methoxy-6-methyl-2-oxo-3-pyridinyl)methyl)-3,4-dihydro-7-((R)-methoxy-3-oxetanylmethyl)-
  • (R)-5,8-dichloro-7-(methoxy(oxetan-3-yl)methyl)-2-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3,4-dihydroisoquinolin-1(2H)-one

Quick Details

  • ProName: PF-06821497
  • CasNo: 1844849-10-0
  • Molecular Formula: C22H24Cl2N2O5
  • Application: For research use only.
  • Purity: 95%
  • LimitNum: 0

Superiority

We provide customized and high-quality PF-06821497 product for your project.

Details

PF-06821497 is a potent, selective and orally active Enhancer of Zeste Homolog 2 (EZH2) inhibitor, with a Ki value <0.1 nM against mutant Y641N EZH2.

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